FIELD: organic chemistry, medicine, oncology, pharmacy. SUBSTANCE: invention relates to novel fluoro-derivative of 1,3,5-oxadiazine eliciting the expressed antitumor effect relative to breast adenocarcinoma cells. Invention describes 2,2,6,6-tetrakis-(trifluoromethyl)-4-ethylamino-5,6-dihydro-1,3,5-oxadiazine of the formula: . Invention proposes also method of its synthesis and pharmaceutical composition based on thereof. Invention provides preparing the novel compound eliciting valuable biological properties. EFFECT: improved method of synthesis, valuable medicinal properties. 3 cl, 1 tbl, 3 ex
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Authors
Dates
2003-05-10—Published
2001-10-12—Filed