TAXANE PENTACYCLIC COMPOUND AND ANTITUMOR AGENTS BASED ON THEREOF Russian patent published in 2005 - IPC

Abstract RU 2257387 C2

FIELD: organic chemistry, medicine, oncology, pharmacy.

SUBSTANCE: invention relates to a new pentacyclic compound derivative of taxane represented by the formula:

wherein R1 represents dimethylaminomethyl group or morpholinomethyl group; R2 represents halogen atom or alkoxy-group comprising from 1 to 6 carbon atoms, or its salt eliciting an antitumor effect, and to a medicine agent based on its. Invention provides preparing new derivatives of taxane eliciting the valuable biological effect.

EFFECT: valuable medicinal properties of compound.

13 cl, 1 dwg, 4 tbl, 16 ex

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RU 2 257 387 C2

Authors

Soga Tsunekhiko

Uoto Kouiti

Takeda Jasujuki

Dates

2005-07-27Published

2000-10-12Filed