APPLYING AGONISTS OF GAMMA-AMINOBUTYRIC ACID RECEPTORS OF B-TYPE AND THEIR PHARMACEUTICALLY ACCEPTABLE DERIVATIVES IN TREATMENT OF NICOTINE DEPENDENCE Russian patent published in 2005 - IPC

Abstract RU 2262352 C2

FIELD: medicine, narcology, pharmacy.

SUBSTANCE: invention proposes applying the following agonists of gamma-aminobutyric acid receptors of B-type: β-(4-chlorophenyl)-GABA (Baclofen), 3-aminopropyl(methyl)-phosphinic acid, 3-aminopropylphosphinic acid, Y-amino-β-4-(4-chlorophenyl)-nitropropane or their salts, esters, ethers, complexes and their corresponding isomers used in treatment of nicotine dependence. Invention provides the selective suppression of smoking addiction and effect on behavior indices causing the abuse relapse and with absence of symptoms typical in nicotine dependence.

EFFECT: valuable properties of compounds.

9 cl

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RU 2 262 352 C2

Authors

Dzhessa Dzhian Luidzhi

Kolombo Dzhiankarlo

Pani Luka

Fratta Val'Ter

Dates

2005-10-20Published

2000-06-30Filed