INHIBITORS OF BACTERIAL GYRASE AND THEIR APPLYING Russian patent published in 2005 - IPC

Abstract RU 2262932 C2

FIELD: organic chemistry, biochemistry, medicine, pharmacology.

SUBSTANCE: invention relates to gyrase inhibitors that reduce amount of microorganisms in biological sample by contacting the indicated sample with compound of the formula (I): , to a method for treatment of bacterial infection by using compounds of the formula (I), compounds of the formula (I) and a pharmaceutical composition comprising compounds of the formula (I). Invention provides the enhanced effectiveness of treatment.

EFFECT: valuable medicinal properties of gyrase.

54 cl, 5 tbl, 13 ex

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RU 2 262 932 C2

Authors

Grijo Ann-Lor

Charifson Pol

Stamos Din

Lajo Jusheng

Badia Majkl

Trjudo Martehn

Dates

2005-10-27—Published

2001-12-12—Filed