FIELD: organic chemistry, medicine, pharmacy.
SUBSTANCE: invention relates to substituted 8,8a-dihydro-3aH-indeno[1,2-d]thiazoles and to their physiologically acceptable salts and physiologically functional derivatives also. Invention describes compounds of the formula (I): 
wherein R1 and R1' mean independently of one another H, F, Cl, Br, J; R2 and R3 means H; R4 means phenyl hat can be replaced with hydroxyl group (OH); R5 means hydrogen atom (H); R6 means OH. Also, invention describes a method for preparing these compounds. Compounds can be used as anorexic agents for prophylaxis and treatment of obesity.
EFFECT: improved preparing method, valuable medicinal properties of compounds.
5 cl, 2 tbl, 1 ex
| Title |
Year |
Author |
Number |
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2001 |
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- Bikkel' Martin
|
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2001 |
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1999 |
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|
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2000 |
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2002 |
- Defossa Ehlizabet
- Klabunde Tomas
- Burger Khans-Jorg
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2001 |
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|
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| DERIVATIVES OF 1,3-DIARYL-2-PYRIDINE-2-YL-3-(PYRIDINE-2-YLAMINO)PROPANOL AND PHARMACEUTICAL COMPOSITION BASED ON THEREOF |
1999 |
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|
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| SUBSTITUTED THIAZOLBENZOISOTHIAZOL DIOXIDE DERIVATIVES, METHOD OF PRODUCTION AND APPLICATION |
2004 |
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|
RU2350613C2 |
