METHOD FOR PREPARING TAXANE DERIVATIVES Russian patent published in 2006 - IPC C07D305/14 C07D493/08

Abstract RU 2275365 C2

FIELD: organic chemistry, chemical technology.

SUBSTANCE: invention relates to a method for preparing derivatives of taxane, namely 13-(N-Boc-β-isobutylisoserinyl)-14-β-hydroxybaccatin III-1,14-carbonate of the formula (I): from 10-desacetylbaccatin III for nine stages. Invention provides the effective method for preparing valuable biologically active compound from the more available parent raw.

EFFECT: improved preparing method.

11 cl, 2 tbl, 8 ex

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RU 2 275 365 C2

Authors

Pontiroli Alessandro

Bombardelli Ehtsio

Dates

2006-04-27—Published

2001-11-22—Filed