ARIPIPRAZOLE MEDICINAL AGENT OF LOW HYGROSCOPICITY AND METHODS FOR ITS PREPARING Russian patent published in 2006 - IPC C07D401/12 A61K31/496 A61P25/18 

Abstract RU 2279429 C2

FIELD: pharmacy.

SUBSTANCE: invention relates to the improved formulation of aripiprazole showing the reduced hygroscopicity. These formulations are not converted to hydrate and not loss the initial solubility being even the medicinal preparation comprising anhydrous apipiprazole crystals are stored for a long time. Also, invention describes method for preparing these formulation and pharmaceutical composition based on thereof.

EFFECT: improved and valuable pharmaceutical properties of agent.

22 cl, 32 dwg, 7 tbl, 28 ex

Similar patents RU2279429C2

Title Year Author Number
LOW HYGROSCOPICITY ARYPYPRAZOLE MEDICINAL AGENT AND METHODS FOR ITS PREPARING 2002
  • Bando Takudzi
  • Aoki Satosi
  • Kavasaki Dzuniti
  • Isigami Makoto
  • Taniguti Jouiti
  • Jabuuti Tsujosi
  • Fudzimoto Kijosi
  • Nisioka Josikhiro
  • Kobajasi Norijuki
  • Fudzimura Tsutomu
  • Takakhasi Masanori
  • Abe Kaoru
  • Nakagava Tomonori
  • Sinkhama Koiti
  • Utsumi Naoto
  • Tominaga Mitiaki
  • Oi Josikhiro
  • Jamada Sokhei
  • Tomikava Kendzi
RU2259366C2
DERIVATIVES OF CARBOSTYRIL AND STABILISERS OF MOOD FOR TREATMENT OF DISORDERS OF MOOD 2004
  • Kikuti Tetsuro
  • Ivamoto Taro
  • Khirose Tsujosi
RU2359675C2
CARBOSTYRIL DERIVATIVES AND SEROTONIN REUPTAKE INHIBITORS FOR PHRENOPATHY TREATMENT 2003
  • Kikuti Tetsuro
  • Ivamoto Taro
  • Khirose Tsujosi
RU2356554C2
CARBOSTYRIL DERIVATIVES AND SEROTONIN REUPTAKE INHIBITORS FOR TREATING PHRENOPATHIES 2008
  • Kikuti Tetsuro
  • Ivamoto Taro
  • Khirose Tsujosi
RU2389490C2
CRYSTALLINE POLYMORPHYL OF 4-[5-(PYRIDINE-4-YL)-1H-1,2,4-TRIAZOL-3-YL]-PYRIDINE-2-CARBONITRILE AND METHOD OF ITS OBTAINING 2013
  • Ivabuti Josiyuki
  • Miyata Satikho
  • Sato Takakhiro
  • Uda Dzunitiro
  • Kandou Takamitsu
  • Inoue Tadasi
  • Nakano Khiroyuki
RU2639149C2
CRYSTALLINE INDOLESULFONAMIDE COMPOUND AND METHOD OF ITS OBTAINING 2004
  • Takakhasi Kejko
  • Khajasi Kendzi
  • Abe Tajti
  • Omae Takao
  • Kato Takasi
RU2336269C2
ALPHA-FORM OR BETA-FORM OF CRYSTAL OF ACETANILIDE DERIVATIVE 2002
  • Kavazoe Souitirou
  • Sakamoto Kenitirou
  • Avamura Judzi
  • Marujama Tatsuja
  • Suzuki Takajuki
  • Onda Keniti
  • Takasu Tosijuki
RU2303033C2
SALT OF PYRROLIDIN-3-YL-ACETIC ACID DERIVATIVE AND ITS CRYSTALS 2014
  • Josida Kensi
  • Kusida Ikuo
RU2640047C2
CRYSTALS OF CYCLIC AMINE DERIVATIVE AND PHARMACEUTICAL USE THEREOF 2017
  • Takahashi Hirozumi
  • Baba Yoko
  • Morita Yasuhiro
  • Iseki Katsuhiko
  • Izumimoto Naoki
RU2719384C1
CRYSTAL FORM OF 4-(3-CHLORINE-4-(CYCLOPROPYLAMINOCARBONYL)AMINOPHENOXY)-7-METHOXY-6-QUINOLINECARBOXAMIDE SALT OR ITS SOLVATE AND METHODS FOR ITS PRODUCING 2004
  • Matsusima Tomokhiro
  • Nakamura Taidzu
  • Josizava Kazukhiro
  • Kamada Atsusi
  • Ajata Jusuke
  • Suzuki Naoko
  • Arimoto Itaru
  • Sakaguti Takakhisa
  • Gotoda Masakharu
RU2328489C2

RU 2 279 429 C2

Authors

Bando Takudzi

Aoki Satosi

Kavasaki Dzuniti

Isigami Makoto

Taniguti Jouiti

Jabuuti Tsujosi

Fudzimoto Kijosi

Nisioka Josikhiro

Kobajasi Norijuki

Fudzimura Tsutomu

Takakhasi Masanori

Abe Kaoru

Nakagava Tomonori

Sinkhama Koiti

Utsumi Naoto

Tominaga Mitiaki

Oi Josikhiro

Jamada Sokhei

Tomikava Kendzi

Dates

2006-07-10Published

2002-09-25Filed