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(19)

(11)

2 304 580

(13)

(51)

IPC

C07D317/62(2006-01-01)

C07D405/12(2006-01-01)

C07D451/06(2006-01-01)

C07D317/46(2006-01-01)

C07D405/14(2006-01-01)

A61K31/36(2006-01-01)

C07D401/06(2006-01-01)

C07D413/06(2006-01-01)

A61P5/02(2006-01-01)

C07D401/12(2006-01-01)

C07D417/06(2006-01-01)

(21) (22)

Application

2005105682/04, 2003-07-18

(24)

Start date

2003-07-18

(22)

Actual filing date

2003-07-18

(45)

Published

2007-08-20

(72)

Inventor

Alanen AleksanderBelajkher KonradGuba Vol'FgangKhap Vol'FgangK'Juber DagmarLjubbers TomasPlanshe Zhan-MarkRozher-Ehvan MarkShnajder GisbertTsjugge JokhenRoshe Oliv'E

(73)

Holder

F.Khoffmann-Lja Rosh Ag

NOVEL BENZODIOXOLS Russian patent published in 2007 - IPC C07D317/62 C07D405/12 C07D451/06 C07D317/46 C07D405/14 A61K31/36 C07D401/06 C07D413/06 A61P5/02 C07D401/12 C07D417/06

Abstract RU 2304580 C2

FIELD: organic chemistry, medicine, pharmacy.

SUBSTANCE: invention relates to novel derivatives of benzodioxol of the formula (I): wherein R¹, R², R³, R⁴, R⁵, R⁶, R⁷ and X are given in the description and the invention claim, and to their pharmaceutically acceptable salts. Also, invention relates to pharmaceutical compositions based on compounds of the formula (I) and their using for preparing medicinal agents used in treatment and/or prophylaxis of diseases associated with modulation of CB1 receptors.

EFFECT: valuable medicinal properties of compounds and pharmaceutical compositions.

19 cl, 279 ex

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RU 2 304 580 C2

Authors

Alanen Aleksander

Belajkher Konrad

Guba Vol'Fgang

Khap Vol'Fgang

K'Juber Dagmar

Ljubbers Tomas

Planshe Zhan-Mark

Rozher-Ehvan Mark

Shnajder Gisbert

Tsjugge Jokhen

Roshe Oliv'E

Dates

2007-08-20—Published

2003-07-18—Filed