3-AMINOPYPERIDINE DERIVATIVES AND METHODS FOR PRODUCTION THEREOF Russian patent published in 2007 - IPC C07D211/56 

Abstract RU 2309147 C9

FIELD: organic chemistry.

SUBSTANCE: invention relates to improved method for production of 3-aminopyperidine derivatives of formula Ib useful in production of protein kinases, wherein R1 is C1-C6-alkyl; R2 is hydrogen, C1-C6-alkyl; R3 is hydrogen, C1-C6-alkyl; R13 is phenyl; n = 1-4. Said method includes reduction of compound of formula II, , wherein R14 is C1-C6-alkyl with reducing agent.

EFFECT: improved method for production of 3-aminopyperidine derivatives.

7 cl, 3 dwg, 2 ex

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RU 2 309 147 C9

Authors

Ripin Dehvid Garol'D Braun

Dates

2007-10-27Published

2003-11-10Filed