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(19)

(11)

2 311 417

(13)

(51)

IPC

C07D495/04(2006-01-01)

C07D487/04(2006-01-01)

A61K31/496(2006-01-01)

A61P15/10(2006-01-01)

A61P15/04(2006-01-01)

(21) (22)

Application

2004101060/04, 2002-08-06

(24)

Start date

2002-08-06

(22)

Actual filing date

2002-08-06

(45)

Published

2007-11-27

(72)

Inventor

Khadson Piter DzheremiPitt Gehri Robert Uil'JamRuker Dejvid FilipBatt Andzhej RomanKhini Selin Margerit SajmonRou Majkl Brajan

(73)

Holder

Ferring Bv

DIAZACYCLOALKANES AS OXYTOCIN AGONISTS Russian patent published in 2007 - IPC C07D495/04 C07D487/04 A61K31/496 A61P15/10 A61P15/04

Abstract RU 2311417 C2

FIELD: organic chemistry, medicine, pharmacy.

SUBSTANCE: invention relates to diazacycloalkanes of the general formula (I): wherein G¹ represents condensed polycyclic group. Compounds are selective and strong acting agonists of oxytocin and can useful in treatment of erectile dysfunction. Also, invention describes a pharmaceutical composition based on compounds of the formula (I) and their using in manufacturing the pharmaceutical composition.

EFFECT: valuable medicinal properties of compounds and pharmaceutical composition.

31 cl, 136 ex

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RU 2 311 417 C2

Authors

Khadson Piter Dzheremi

Pitt Gehri Robert Uil'Jam

Ruker Dejvid Filip

Batt Andzhej Roman

Khini Selin Margerit Sajmon

Rou Majkl Brajan

Dates

2007-11-27—Published

2002-08-06—Filed