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(19)

(11)

2 370 497

(13)

(51)

IPC

C07D487/04(2006-01-01)

C07D267/14(2006-01-01)

C07D265/36(2006-01-01)

C07D215/08(2006-01-01)

C07D498/14(2006-01-01)

C07D513/14(2006-01-01)

C07D417/10(2006-01-01)

C07D231/38(2006-01-01)

C07D267/16(2006-01-01)

C07D333/44(2006-01-01)

C07D223/16(2006-01-01)

A61K31/55(2006-01-01)

A61K31/553(2006-01-01)

A61K31/5517(2006-01-01)

A61K31/495(2006-01-01)

A61K31/38(2006-01-01)

A61P9/04(2006-01-01)

A61P9/12(2006-01-01)

A61P25/24(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2007101239/04, 2005-08-24

(24)

Start date

2005-08-24

(22)

Actual filing date

2005-08-24

(45)

Published

2009-10-20

(72)

Inventor

Andzhej Roman BattBakster Ehndrju DzhonKhini SelinStokli Martin LiBrajan Ro MajklKhadson PiterKhehndi Rejchel

(73)

Holder

Vantia Limited

VASOPRESSIN V RECEPTOR ANTAGONISTS Russian patent published in 2009 - IPC C07D487/04 C07D267/14 C07D265/36 C07D215/08 C07D498/14 C07D513/14 C07D417/10 C07D231/38 C07D267/16 C07D333/44 C07D223/16 A61K31/55 A61K31/553 A61K31/5517 A61K31/495 A61K31/38 A61P9/04 A61P9/12 A61P25/24 A61P35/00

Abstract RU 2370497 C2

FIELD: pharmacology.

SUBSTANCE: invention concerns novel compounds of formula (1a), formula (1b), formula (1c) and formula (1d), as well as pharmaceutical composition based on them and their application in medicine obtainment. R¹-R⁴, G, W, X, X¹, U, V, a, b are defined in the invention claim.

EFFECT: compound with antagonistic effect on vasopressin V1A receptor.

73 cl, 133 ex

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RU 2 370 497 C2

Authors

Andzhej Roman Batt

Bakster Ehndrju Dzhon

Khini Selin

Stokli Martin Li

Brajan Ro Majkl

Khadson Piter

Khehndi Rejchel

Dates

2009-10-20—Published

2005-08-24—Filed