ACID INSULIN PREPARATIONS WITH ENHANCED STABILITY Russian patent published in 2007 - IPC A61K38/28 A61P3/10 

Abstract RU 2313362 C2

FIELD: chemical-pharmaceutical industry, pharmacy.

SUBSTANCE: invention relates to a composition comprising Gly(A21),Arg(B31),Arg(B32)-human insulin, at least one chemical substance chosen from polyatomic alcohols and their ester and ethers, at least one preserving agent and water wherein pH of this pharmaceutical composition is in acid region (pH 1-6.8). The claimed composition possesses the enhanced stability and resistance against aggregation in storage, prolonged effect period that provides administration of the claimed composition once for 24 h.

EFFECT: improved, enhanced and valuable properties of preparations.

23 cl, 11 tbl, 3 ex

Similar patents RU2313362C2

Title Year Author Number
ZINC-FREE AND ZINC-DEPLETED INSULIN COMPOSITIONS OF INCREASED STABILITY 2002
  • Boderke Peter
RU2311922C2
INSULIN PREPARATION CONTAINING METHIONINE 2010
  • Shettle Izabell'
  • Khagendorf Annika
  • Fjurst Kristiane
  • Khauk Gerrit
  • Zifke-Khentsler Ferena
  • Kamm Val'Ter
  • Shniders Julija
RU2540485C2
PHARMACEUTICAL COMPOSITION CONTAINING AGONIST GLP-1, INSULIN AND METHIONINE 2010
  • Khagendorf Annika
  • Khauk Gerrit
  • Mjuller Verner
  • Shettle Izabell'
  • Zifke-Khentsler Ferena
  • Terch Katrin
RU2537239C2
COMBINATION OF INSULIN AND GLP-1 AGONIST 2014
  • Verner Ulrikh
  • Rottkhojzer Berbel
  • Smit Kristofer Dzhejms
RU2682671C2
NOVEL INSULIN DERIVATIVES WITH STRONGLY SLOWED PROFILE TIME/ACTION 2009
  • Khabermann,Paul'
  • Zajpke,Gerkhard
  • Kurrle,Roland
  • Mjuller,Gjunter
  • Zommerfel'D,Mark
  • Tennagel'S,Norbert
  • Chank,Georg
  • Verner,Ul'Rikh
RU2529952C2
COMBINATION OF INSULIN AND GLP-1 AGONIST 2009
  • Verner Ul'Rikh
  • Rottkhojzer Berbel'
  • Smit Kristofer Dzhejms
RU2532378C2
ACYLATED INSULIN ANALOGUES STABILISED WITH RESPECT TO PROTEASES 2009
  • Madsen Peter
  • K'El'Dsen Tomas Berglum
  • Khoeg-Jensen Tomas
  • Jakobsen Palle
  • Tagmose Tina Meller
  • Glendorf Tine
  • Kodra Janosh Tibor
  • Gehribehj Patrik Uill'Jam
  • Petersen Jakob Sten
RU2571857C2
NOVEL INSULIN DERIVATIVES WITH EXTREMELY DELAYED TIME/ACTION PROFILE 2009
  • Khabermann Paul'
  • Zajpke Gerkhard
  • Kurrle Roland
  • Mjuller Gjunter
  • Zommerfel'D Mark
  • Tennagel'S Norbert
  • Chank Georg
  • Verner Ul'Rikh
RU2524423C2
STRAIN OF ESCHERICHIA COLI BACTERIA WITH REDUCED ABILITY TO ACCUMULATE ACETATE - PRODUCER OF HYBRID POLYPEPTIDE CONTAINING PROINSULIN GLARGINE 2023
  • Rodionov Petr Petrovich
  • Latypov Vitalii Feliksovich
  • Selivanova Tatiana Aleksandrovna
RU2807548C1
STABLE NON-AQUEOUS PHARMACEUTICAL COMPOSITIONS 2008
  • B'Erregord Jensen Simon
  • Khavelund Svend
  • Feger Florian Anders
RU2472492C2

RU 2 313 362 C2

Authors

Brunner-Shvarts Anette

Lill' Norbert

Dates

2007-12-27Published

2003-06-05Filed