USE OF NOVEL ETHONOGESTREL ESTERS Russian patent published in 2008 - IPC A61K31/568 A61P15/00 

Abstract RU 2322986 C2

FIELD: medicine, steroids, pharmacy.

SUBSTANCE: invention describes a pharmaceutical composition based on oil for injection contraception and/or for substitution hormonal therapy. The composition comprises the effective amount of ethonogestrel decanoate and/or ethonogestrel undecanoate, and/or ethonogestrel dodecanoate taken in the effective contraception and/or therapeutic acting doses. Also, invention describes a method for carrying out the contraception and/or substitution hormonal therapy. Use of specific ethonogestrel esters provides good pharmacokinetic pattern and gives the possibility for using progestogen in a single dose with the prolonged period of effect.

EFFECT: improved and valuable medicinal and pharmaceutical properties of compounds.

10 cl, 2 tbl, 6 dwg, 4 ex

Similar patents RU2322986C2

Title Year Author Number
CONTRACEPTIVE INJECTION OF OIL SOLUTION INJECTED INDEPENDENTLY 2003
  • De Nejs Khenrik
  • Van Der Vort Khendrikus Adrianus Antonius
  • Lejsen Dirk
RU2328289C2
NEW ESTERS OF ETHONOGESTREL 2003
  • De Nejs Khenrik
  • Van Der Vort Khendrikus Adrianus Antonius
  • Lejsen Dirk
  • Grotenkhejs Arej Jan
RU2325910C2
STEROIDS WITH MIXED ANDROGENIC AND PROGESTAGENIC PROFILE 2004
  • Van Der Lou Jap
  • Lejsen Dirk
  • Grotenkhejs Arej Jan
  • De Gojer Marsel' Ehvert
RU2357972C2
COMPOUND (α)-7-METHYL-17-[(1-OXOUNDECYL)OXY]-ESTR-4-ENE-3-ONE, PHARMACEUTICAL COMPOSITION, SET FOR MALE CONTRACEPTION 1999
  • Lejsen Dirk
  • Van Der Vort Khendrikus Adrianus Antonius
RU2216546C2
COMPOUNDS, SET, ANDROGENIC COMPOSITION 2000
  • Lejsen Dirk
  • Van Der Lau Jap
  • Buma Bursi Roberta
  • De Gojer Marsel' Ehvert
RU2242479C2
METHOD AND PHARMACEUTICAL COMPOSITIONS FOR RELIABLE ACHIEVEMENT OF ACCEPTABLE LEVELS OF TESTOSTERONE IN SERUM 2004
  • Khjubler Doris
  • Frikke Zabine
  • Ingverzen Jan-Peter
  • Kunts Vil'Khel'M
RU2354381C2
STEROID COMPOUND, ITS USING AND TREATMENT METHOD 2002
  • Van Der Lau Jap
  • Lejsen Dirk
  • De Gojer Marsel Ehvert
RU2294332C2
METHOD FOR PREPARING 7α-METHYLSTEROIDS, COMPOUND 2003
  • Stulvinder J.
  • Ostendorf M.
  • Bjugenjum Van P.A.M.
RU2305105C2
INDOLES USEFUL IN TREATMENT ANDROGEN RECEPTORS BOUND DESEASES 2003
  • Khermkens Pedro Kharol'D Khan
  • Stok Kherman Tejs
  • Terkhejs Nel'T'E Miranda
  • Lommerse Jokhannes Petrus Marija
  • Van Der Lou Jap
RU2328484C2
HORMONAL OR ANTI-HORMONAL STEROID COMPOUNDS, METHODS FOR THERAPEUTIC EFFECT, METHOD FOR PREPARING COMPOUNDS 1999
  • Kuk K. Ehdgar
  • Kepler Dzhon A.
  • Bartli Gari S.
  • Shetti Rupa S.
RU2238943C2

RU 2 322 986 C2

Authors

De Nejs Khenrik

Van Der Vort Khendrikus Adrianus Antonius

Lejsen Dirk

Grotenkhejs Arej Jan

Van Der Lou Jap

Dates

2008-04-27Published

2003-05-22Filed