STEROIDS WITH MIXED ANDROGENIC AND PROGESTAGENIC PROFILE Russian patent published in 2009 - IPC C07J63/00 A61K31/56 A61P5/26 A61P5/34 

Abstract RU 2357972 C2

FIELD: medicine.

SUBSTANCE: invention claims 19-nor-D-homosteroids with mixed androgenic/progestagenic profile and oral activity, preventing bone mineral density (BMD) loss in trabecular bones, with zero liver toxicity, with structure of the formula (I) , where R1 is O, R2 is methyl or ethyl, and R3 is hydrogen.

EFFECT: improved efficiency of composition and treatment method.

9 cl, 3 ex, 3 tbl

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RU 2 357 972 C2

Authors

Van Der Lou Jap

Lejsen Dirk

Grotenkhejs Arej Jan

De Gojer Marsel' Ehvert

Dates

2009-06-10Published

2004-12-15Filed