METHOD OF 2-SULPHONILAMINE-1,2,4,-TRIAZOLO[1,5-a] PYRIMIDINES PRODUCTION Russian patent published in 2008 - IPC C07D487/04 

Abstract RU 2325390 C1

FIELD: chemistry.

SUBSTANCE: invention refers to organic substances production and can be applied for production of herbicides and other bioactive compounds. Production of 2-sulphanilamine-1,2,4-triazolo[1,5-a]pyrimidine of general formula , where R1 is metal, phenylic, 4-methyl phenylic, 4-chlorophenylic group, R is phenylic, 4-methyl phenylic, 4-chlorophenylic, methoxyphenylic group, R is metal, phenylic, 4-methyl phenylic, 4-chlorophenylic group is sulphurization of 2-amino-4,7-dihydro-1,2,4-triazolo [1,5-a]pyrimidines (II) by sulphochlorides (III) in pyrimidine and oxidation of produced 2-sulphanilamine-4,7-dihydro-1,2,4-triazolo[1,5-a] pyrimidines (IV) by bromine in acetic acid with sodium acetate occurrence.

EFFECT: method allows to produce compounds using low-price and reasonable raw materials without any complicated processing steps applied.

1 cl, 7 ex

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RU 2 325 390 C1

Authors

Chernyshev Viktor Mikhajlovich

Sokolov Andrej Nikolaevich

Taranushich Vitalij Andreevich

Dates

2008-05-27Published

2007-01-29Filed