2-(5-NITRONYLFURAN-2-YL)-5-METHYL-6-NITRO-1,2,4-TRIAZOLO[1,5-A]PYRIMIDIN-7(4N)-ONE AND SALTS THEREOF Russian patent published in 2020 - IPC C07D487/04 A61K31/519 A61P9/10 A61P9/04 A61P3/10 

Abstract RU 2716715 C2

FIELD: medicine.

SUBSTANCE: invention relates to 2-(5-nitronylfuran-2-yl)-methyl-6-nitro-1,2,4-triazolo[1,5-a]pyrimidin-7-one (2a-z).

EFFECT: obtaining novel compounds which exhibit an antiglycating and inhibitory effect on α-glucosidase activity, which can be used in medicine for treating and preventing the consequences of diabetes mellitus.

1 cl, 3 tbl, 11 ex

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Authors

Chupakhin Oleg Nikolaevich

Charushin Valerij Nikolaevich

Rusinov Vladimir Leonidovich

Savateev Konstantin Valerevich

Ulomskij Evgenij Nartsissovich

Fedotov Viktor Vladimirovich

Petrov Vladimir Ivanovich

Spasov Aleksandr Alekseevich

Babkova Valentina Andreevna

Babkov Denis Aleksandrovich

Dates

2020-03-16Published

2018-07-30Filed