FIELD: chemistry.
SUBSTANCE: described is novel compound of formula (I)
or its pharmaceutically acceptable salt, values of radicals are given in invention formula Compound has ability to inhibit receptor mGluR5, which intends it for prevention and/or treatment of receptor mGluR5- associated disturbances. Also described is pharmaceutical composition, method of inhibiting activation of receptors mGluR5, using compound of formula (I). Described is method of obtaining compound of formula 1a or 1b structure.
EFFECT: increasing output of suitable product.
18 cl, 825 ex
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Authors
Dates
2009-04-20—Published
2003-08-08—Filed