1-(2-AMINOBENZOL)PIPERAZINE DERIVATIVES AS GLYCIN UPTAKE INHIBITORS TO BE USED FOR PSYCHOSIS TREATMENT Russian patent published in 2009 - IPC C07D295/192 C07D401/10 C07D403/10 C07D403/12 C07D403/14 C07D417/10 C07D417/14 A61K31/496 A61K31/495 A61P25/28 

Abstract RU 2354653 C2

FIELD: chemistry.

SUBSTANCE: there are disclosed 1-(2-aminobenzol)piperazine derivatives of formula (I) and pharmaceutically acceptable acid-additive salts with radical values specified in patent claim. The compounds are characterised with inhibiting effect on glycine I carrier. There is also disclosed medical product based on the compounds of formula (I).

EFFECT: compound can be used for treatment of the diseases associated with glycine uptake inhibition.

12 cl, 5 tbl, 396 ex

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RU 2 354 653 C2

Authors

Al'Berati-Dzhiani Daniela

Kholidon Sinese

Narkizjan Rober

Nettekoven Mattias Genrikh

Norkross Rodzher Dejvid

Pinar Ehmman'Juehl'

Shtadler Khenri

Dates

2009-05-10Published

2004-08-30Filed