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(19)

(11)

2 443 706

(13)

(51)

IPC

C07D491/04(2006-01-01)

C07D495/04(2006-01-01)

C07D519/00(2006-01-01)

A61K31/5025(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2008145660/04, 2007-04-24

(24)

Start date

2007-04-24

(22)

Actual filing date

2007-04-24

(45)

Published

2012-02-27

(72)

Inventor

Folks EhdrianShattlvort StefenChakovri IrinaOksenford SalliVan Nan ChiKastanedo DzhordzhettaGanzner DzhenetKheffron TimMat'E SimonOlivero AlanSazerlin Dehniel' P.Chzhu Bin-Jan'Goldsmit Richard

(73)

Holder

Dzhenentek, Ink.F. Khoffmann-Lja Rosh Ag

PHARMACEUTICAL COMPOUNDS Russian patent published in 2012 - IPC C07D491/04 C07D495/04 C07D519/00 A61K31/5025 A61P35/00

Abstract RU 2443706 C2

FIELD: chemistry.

SUBSTANCE: invention relates to compounds of formulae

and ,

which can be used to inhibit lipid kinase, including PI3K, and treat lipid kinase-mediated disorders. Values of radicals are given in claim 1.

EFFECT: improved properties of the compound.

11 cl, 2 tbl, 7 ex

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RU 2 443 706 C2

Authors

Folks Ehdrian

Shattlvort Stefen

Chakovri Irina

Oksenford Salli

Van Nan Chi

Kastanedo Dzhordzhetta

Ganzner Dzhenet

Kheffron Tim

Mat'E Simon

Olivero Alan

Sazerlin Dehniel' P.

Chzhu Bin-Jan'

Goldsmit Richard

Dates

2012-02-27—Published

2007-04-24—Filed