15β-SUBSTITUTED STEROIDS WITH SELECTIVE OESTROGENIC ACTIVITY Russian patent published in 2010 - IPC C07J1/00 A61P5/00 A61K31/56 

Abstract RU 2386637 C2

FIELD: chemistry.

SUBSTANCE: described is a 15β-substituted oestradio derivative having selective oestrogenic activity. The preferred compound is 7α-ethyl-15β-methyl-19-nor-17α-pregna-1,3,5(10)-trien-20-yne-3,17β-diol.

EFFECT: obtaining compounds which can be used in treating or preventing diseases or physiological conditions related to oestrogen receptors.

11 cl, 4 ex, 2 tbl

Similar patents RU2386637C2

Title Year Author Number
STEROID COMPOUNDS, METHOD FOR SELECTIVE MODIFICATION, PHARMACEUTICAL COMPOSITION 2001
  • Lozen Khjubert Jan Jozef
RU2255090C2
COMPOUNDS, SET, ANDROGENIC COMPOSITION 2000
  • Lejsen Dirk
  • Van Der Lau Jap
  • Buma Bursi Roberta
  • De Gojer Marsel' Ehvert
RU2242479C2
15,15-DIALKYLSTEROID COMPOUNDS AND METHOD OF PREPARATION THEREOF 1994
  • Dzhejms Ronal'D Ball
  • Karl-Khajnrikh Frittsemajer
  • Krista Khegele-Khartung
RU2147306C1
PROGESTERONE RECEPTOR MODULATORS 2005
  • Khamersma Jokhannes Antonius Marija
  • Revinkel Jokhannes Bernardus Marija
RU2381232C2
NONAROMATIC ESTROGENIC STEROID, PHARMACEUTICAL COMPOSITION 2000
  • Lozen Khjubert Jan Jozef
  • Veneman Gerrit Kherman
  • Skhonen Vil'Khel'Mus Gerardus Ehduardus Josef
RU2245886C2
BRIDGE-CONTAINING ESTRATRIENES 1990
  • Geral'D Kirsh[De]
  • Gjunter Neef[De]
  • Khenri Laurent[De]
  • Rudol'F Vikhert[De]
  • Dzhejms R.Ball[Za]
  • Peter Ehsperling[De]
  • Val'Ter Ehl'Ger[De]
  • Sjubille Bajer[De]
RU2087479C1
METHOD OF SYNTHESIS OF SULFATIZED ESTROGEN MIXTURE 1998
  • Rajmakers Petrus Khendrikus
  • Khofstrat Robert Gerrit
  • Bom Khenrikus Petrus Antonius Jokhannes Marija Van Den
RU2184741C2
18-METHYL-19-NORANDROST-4-ENE-17,17-SPIROETHER (18-METHYL-19-NOR-20-SPIROX-4-EN-3-ON) AND PHARMACEUTICAL PREPARATIONS CONTAINING SAID COMPOUND 2007
  • Bol'Mann Rol'F
  • Kunke Joakhim
  • Khjubner Jan
  • Gallus Norbert
  • Menges Frederik
  • Borden Shteffen
  • Mun Khans-Peter
  • Prelle Katja
RU2440365C2
SULFAMATE DERIVATIVES, METHOD OF PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITIONS 1996
  • Zigfrid Shvarts
  • Val'Ter Ehl'Ger
  • Gudrun Reddersen
  • Birgitt Shnajder
  • Ina Time
  • Margit Rikhter
RU2159774C2
DERIVATIVES OF 11,21-BISPHENYL-19-NORPREGNANE, METHOD OF THEIR SYNTHESIS, PHARMACEUTICAL COMPOSITION AND METHOD OF ITS PREPARING 1995
  • Gebkhar Ronal'D
  • Van Der Vort Khendrikus Adrianus Antonius
RU2152952C2

RU 2 386 637 C2

Authors

Lozen Khubert Jan Jozef

Ehderven Antonius Gerardus Khendrikus

Dejks Frederikus Antonius

Dates

2010-04-20Published

2005-09-05Filed