INDOLYLMALEIMIDE DERIVATIVES Russian patent published in 2009 - IPC C07D403/04 A61K31/404 

Abstract RU 2373201 C2

FIELD: chemistry.

SUBSTANCE: invention relates to new indolylmaleimide derivatives of formula I: , where: Ra is H, C1-4alkyl; one of Ra, Rc, Rd and Re is C1-4alkyl; and the other three substitutes are H; or Rb, Rd, Re are all H; and R is a radical of formula (a): , where R1 is -(CH2)n-NR3R4, where each of R3 and R4 are independently H, C1-4alkyl; n is 0, 1, 2; R2 is H; halogen; or its pharmaceutically acceptable salt.

EFFECT: wider field of use of the compounds.

8 cl, 1 tbl, 1 ex

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RU 2 373 201 C2

Authors

Van-Ehjs Mauris

Fon-Matt Peter

Vagner Jurgen

Ehvenu Zhan-P'Err

Dates

2009-11-20Published

2005-01-19Filed