NEW BLOCK COPOLYMER, MICELLAR PREPARATION AND ANTICARCINOGENIC AGENT CONTAINING MICELLAR PREPARATION AS ACTIVE COMPONENT Russian patent published in 2009 - IPC C08G69/40 A61K9/107 A61K31/337 A61K45/00 A61K47/34 

Abstract RU 2375384 C2

FIELD: medicine.

SUBSTANCE: block copolymer is produced by reaction of a compound containing a structure fragment of polyethylene glycol and a structure fragment of polyamino acid in a solvent at temperature 30 to 60°C within 2-48 hours. The prepared block copolymer is used as a carrier for an anticarcinogenic taxtane agent, particularly Paclitaxel in a micellar preparation in amount required for disease treatment.

EFFECT: ensured absence of allergic reaction, higher solubility of the sparingly water-soluble anticarcinogenic agent, maintained high blood concentration of the medicine, accumulation of high concentration of the medicine in tumour tissue, intensified pharmacological action and decrease in by-effects.

13 cl, 6 tbl, 4 ex

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RU 2 375 384 C2

Authors

Simizu Kazukhisa

Isikava Kejzou

Nakanisi Takesi

Dates

2009-12-10Published

2005-09-16Filed