4-CYCLOALKYL-SUBSTITUTED DERIVATIVES OF TETRAHYDROQUINOLINE AND USE THEREOF AS MEDICINE Russian patent published in 2010 - IPC C07D215/20 

Abstract RU 2393151 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a novel derivative of tetrahydroquinoline of formula (1a) , in which R denotes cyclopentyl or isopropyl, as well as salts, solvate and salt solvates thereof.

EFFECT: novel compounds which can be used as a cholesterol ester transfer protein (CETP) inhibitor are obtained and described.

1 cl, 6 ex

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RU 2 393 151 C2

Authors

Bishoff Khil'Mar

Gilen-Khehrtvig Khajke

Li Fol'Kkhart

Shmek Karsten

Tutevol' Mikhaehl'

Vakolopulos Aleksandros

Veber Olaf

Vuttke Martina

Dates

2010-06-27Published

2005-12-15Filed