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(19)

(11)

2 470 932

(13)

(51)

IPC

C07D471/04(2006-01-01)

A61K31/4375(2006-01-01)

A61P5/42(2006-01-01)

A61P9/04(2006-01-01)

A61P9/10(2006-01-01)

A61P9/12(2006-01-01)

A61P13/12(2006-01-01)

(21) (22)

Application

2009135659/04, 2008-02-19

(24)

Start date

2008-02-19

(22)

Actual filing date

2008-02-19

(45)

Published

2012-12-27

(72)

Inventor

Behrfakker LarsKol'Kkhof PeterShlemmer Karl-KhajntsGrosser Rol'FNitshe AdamKljajn MartinaMjunter KlausAl'Brekht-Kjupper BarbaraKhartmann Ehl'Ke

(73)

Holder

Bajer Shering Farma Aktsiengezel'Shaft

SUBSTITUTED 4-ARYL-1,4-DIHYDRO-1,6-NAPHTHYRIDINE AMIDES AND USE THEREOF Russian patent published in 2012 - IPC C07D471/04 A61K31/4375 A61P5/42 A61P9/04 A61P9/10 A61P9/12 A61P13/12

Abstract RU 2470932 C9

FIELD: chemistry.

SUBSTANCE: invention relates to novel substituted 4-aryl-1,4-dihydro-1,6-naphthyridine-3-carboxamides, method for production thereof, use thereof to produce a medicinal agent which inhibits MR activity.

EFFECT: improved method.

11 cl, 9 ex

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RU 2 470 932 C9

Authors

Behrfakker Lars

Kol'Kkhof Peter

Shlemmer Karl-Khajnts

Grosser Rol'F

Nitshe Adam

Kljajn Martina

Mjunter Klaus

Al'Brekht-Kjupper Barbara

Khartmann Ehl'Ke

Dates

2012-12-27—Published

2008-02-19—Filed