SULFONAMIDE PERI-SUBSTITUTED BICYCLES FOR TREATMENT OF OCCLUSIVE AFFECTION OF ARTERIES Russian patent published in 2010 - IPC C07D209/12 C07D209/30 C07D209/34 C07D401/12 C07D409/12 C07D409/14 C07D413/12 C07D487/04 C07D513/04 A61K31/404 A61K31/416 A61K31/4162 A61P9/10 

Abstract RU 2403240 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: there are described novel acylsulfonamide peri-substituted condensed bicyclic compounds of general formula (I), values of radicals are given in invention formula. Also described is pharmaceutical composition based on formula (I) compound.

EFFECT: compounds can be used for inhibition of prostaglandin E2 binding with receptor EP3.

30 cl, 371 ex, 4 tbl

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RU 2 403 240 C2

Authors

Chzhou Nian'

Singkh Dzhasbir

Garni Mark

Khejtgan Dzhordzheta

Juj Pehn

Zembauehr Dehvid

Dates

2010-11-10Published

2005-06-27Filed