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2 404 179

(13)

(51)

IPC

C07D451/04(2006-01-01)

A61K31/46(2006-01-01)

A61P1/00(2006-01-01)

(21) (22)

Application

2007128061/04, 2005-12-21

(24)

Start date

2005-12-21

(22)

Actual filing date

2005-12-21

(45)

Published

2010-11-20

(72)

Inventor

Fazeri Pol R.Gendron RolandGoldblum AdamLong DehnielMarkess DehnielTerner Derek S.Choj Seok-Ki

(73)

Holder

Terevans, Ink.

INDAZOLE-CARBOXAMIDE COMPOUNDS Russian patent published in 2010 - IPC C07D451/04 A61K31/46 A61P1/00

Abstract RU 2404179 C2

FIELD: chemistry.

SUBSTANCE: invention relates to novel indazole-carboxamide compounds of formula ,

in which radicals and groups are as defined in claim 1 of the formula of invention. Present invention also relates to pharmaceutical compositions containing said compounds, to methods of using such compounds to treat 5-HT₄-receptor mediated diseases.

EFFECT: said compounds are 5-HT₄-receptor agonists.

16 cl, 10 tbl, 21 ex

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RU 2 404 179 C2

Authors

Fazeri Pol R.

Gendron Roland

Goldblum Adam

Long Dehniel

Markess Dehniel

Terner Derek S.

Choj Seok-Ki

Dates

2010-11-20—Published

2005-12-21—Filed