FIELD: chemistry.
SUBSTANCE: invention relates to novel compounds of formula (I): 
where: X denotes -CH2-, -CH2CH2-; R1 denotes H; R2 and R3 denote H; or one of them denotes H and the other denotes a branched or straight C1-6alkyl, C3-6cycloalkyl or phenyl; where the said C1-6alkyl is possibly substituted with one OH, NH2, C3-6cycloalkyl, phenyl; where any phenyl is possibly substituted with one or two substitutes selected from halogen or C1-6alkyl; R4 denotes H; R5 denotes H, halogen, C1-6alkyl; or a pharmaceutically acceptable salt thereof.
EFFECT: compounds inhibit cholesterol absorption, which enables their use in treating and preventing atherosclerosis.
14 cl, 18 ex
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