FIELD: chemistry.
SUBSTANCE: invention relates to tetrahydroquinoline derivatives of formula (I), where values of C3-C4, R2, R3, R4, R5, L1, L2, Y and X are given in claim 1, as muscarinic receptor agonists; compositions containing said compounds; methods of inhibiting muscarinic receptor activity using said compounds; methods of treating diseased conditions associated with the muscarinic receptor using said compounds, and methods of identifying a subject suitable for treatment using said compounds.
EFFECT: improved properties of compounds.
22 cl, 1 tbl, 3 ex, 3 dwg
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Authors
Dates
2011-11-27—Published
2005-12-15—Filed