STABLE SOLID DISPERSION OF VINCA ALKALOID DERIVATIVE AND METHOD FOR PRODUCING THEREOF Russian patent published in 2011 - IPC A61K8/04 A61K9/16 A61K9/48 A61K31/4375 

Abstract RU 2412687 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to pharmacology and medicine, and represents a solid and stable oral dispersion of water-soluble Vinca alkaloid derivative, particularly vinorelbine in at least one polyethylene glycol of molecular weight within 1000 and 6000, wherein a mass ratio of water-soluble vinorelbine and more specifically, firstly vinorelbine ditartrate and, secondly polyethylene glycol is within 1.5:1 and 1:10 and, preferentially within 1:3 and 1:6.

EFFECT: invention provides higher stability of Vinca alkaloid derivatives, and especially vinorelbine salts, particularly vinorelbine ditartrate.

14 cl, 3 ex, 2 tbl, 2 dwg

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RU 2 412 687 C2

Authors

Bugare Zhoehl'

Lever Ehli

Ibarra Mari-Dominik

Dates

2011-02-27Published

2005-12-20Filed