METHOD OF PRODUCING N-[3-[(2-METHOXYPHENYL)SULFANYL]-2-METHYLPROPYL]-3,4-DIHYDRO-2H-1,5- BENZOXATHIEPIN-3-AMINE Russian patent published in 2011 - IPC C07D327/02 C07C323/20 

Abstract RU 2414464 C9

FIELD: chemistry.

SUBSTANCE: invention relates to a method of producing N-[3-[(2-methoxyphenyl)sulfanyl]-2-methylpropyl]-3,4-dihydro-2H-1,5-benzoxathiepin-3-amine of general formula (1) , involving condensation of intermediate compounds of formulae (2) and (3), where R denotes methyl or preferably 4-methylphenyl. The invention also relates to novel compounds of formulae (3), which are used as intermediate compounds in synthesis of formula (1) compounds.

EFFECT: novel method of producing the said compound is safe and cheap.

7 cl, 2 ex

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RU 2 414 464 C9

Authors

Vashe Bernar

Brjunel' Iv

Morel' Zhan-Lui

Dates

2011-03-20Published

2007-11-06Filed