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2 415 128

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IPC

C07C233/65(2006-01-01)

C07D295/03(2006-01-01)

A61K31/452(2006-01-01)

A61P9/00(2006-01-01)

A61P9/06(2006-01-01)

(21) (22)

Application

2009117328/04, 2009-05-07

(24)

Start date

2009-05-07

(22)

Actual filing date

2009-05-07

(45)

Published

2011-03-27

(72)

Inventor

Glushkov Robert GeorgievichJuzhakov Sergej DanilovichDavydova Nadezhda KonstantinovnaZhikhareva Galina PetrovnaRozenshtraukh Leonid ValentinovichGolitsyn Sergej PavlovichSokolov Sergej Fedorovich

(73)

Holder

Obshchestvo S Ogranichennoj Otvetstvennost'Ju Po Khimii Lekarstvennykh Sredstv"Federal'Noe Gosudarstvennoe Uchrezhdenie Kardiologicheskij Nauchno-Proizvodstvennyj Kompleks" Ministerstva Zdravookhranenija I Sotsial'Nogo Razvitija Rossijskoj Federatsii Rknpk Minzdravsotsrazvitija Rossii)

N-1-[(4-FLUOROPHENYL)-2-(1-ETHYL-4-PIPERIDYL)-ETHYL]-4-NITROBENZAMIDE HYDROCHLORIDE EXHIBITING ANTIARHYTHMIC AND ANTIFIBRILLATORY ACTIVITY Russian patent published in 2011 - IPC C07C233/65 C07D295/03 A61K31/452 A61P9/00 A61P9/06

Abstract RU 2415128 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to a new chemical compound - N-1-[(4-fluorophenyl)-2-(1-ethyl-4-piperidyl)-ethyl]-4-nitrobenzamide hydrochloride of formula Also, the invention refers to drugs.

EFFECT: preparation of a new biologically active compound which exhibits antiarhythmic and antifibrillatory activity.

2 cl, 1 ex, 2 tbl

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RU 2 415 128 C2

Authors

Glushkov Robert Georgievich

Juzhakov Sergej Danilovich

Davydova Nadezhda Konstantinovna

Zhikhareva Galina Petrovna

Rozenshtraukh Leonid Valentinovich

Golitsyn Sergej Pavlovich

Sokolov Sergej Fedorovich

Dates

2011-03-27—Published

2009-05-07—Filed