FIELD: medicine, pharmaceutics.
SUBSTANCE: invention refers to new arylamidine derivatives presented by general formula, or to their salts: [Formula 1] where R1 and R2 either identically or differently represent optionally substituted C3-4 alkyl group. Also, the invention refers to 4-{3-[4-(3-{4-[amino(propoxycarbonylimino)methyl]phenoxy}propyl)-1-piperidinyl]propoxy}-N'-(propoxycarbonyl)benzamidine, to 4-{3-[4-(3-{4-[amino(isopropoxycarbonylimino)methyl]phenoxy}propyl)-1-piperidinyl]propoxy}-N'-(isopropoxycarbonyl)benzamidine, to 4-{3-[4-(3-{4-[amino(butoxycarbonylimino)methyl]phenoxy}propyl)-1-piperidinyl]propoxy}-N'-(butoxycarbonyl)benzamidine, as well as to an antifungal agent.
EFFECT: preparation of new biologically active compounds which exhibit antifungal activity.
6 cl, 4 ex
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Authors
Dates
2011-04-10—Published
2006-12-27—Filed