NEW ARYLAMIDINE DERIVATIVE, ITS SALT AND ANTIFUNGAL AGENT CONTAINING IT Russian patent published in 2011 - IPC C07D211/22 A61K31/445 A61P31/10 

Abstract RU 2415839 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to new arylamidine derivatives presented by general formula, or to their salts: [Formula 1] where R1 and R2 either identically or differently represent optionally substituted C3-4 alkyl group. Also, the invention refers to 4-{3-[4-(3-{4-[amino(propoxycarbonylimino)methyl]phenoxy}propyl)-1-piperidinyl]propoxy}-N'-(propoxycarbonyl)benzamidine, to 4-{3-[4-(3-{4-[amino(isopropoxycarbonylimino)methyl]phenoxy}propyl)-1-piperidinyl]propoxy}-N'-(isopropoxycarbonyl)benzamidine, to 4-{3-[4-(3-{4-[amino(butoxycarbonylimino)methyl]phenoxy}propyl)-1-piperidinyl]propoxy}-N'-(butoxycarbonyl)benzamidine, as well as to an antifungal agent.

EFFECT: preparation of new biologically active compounds which exhibit antifungal activity.

6 cl, 4 ex

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RU 2 415 839 C2

Authors

Khajasi Kazuja

Dates

2011-04-10Published

2006-12-27Filed