Show metadata Hide metadata

(19)

(11)

2 299 195

(13)

(51)

IPC

C07C257/18(2006-01-01)

C07D241/08(2006-01-01)

A61K31/155(2006-01-01)

A61K31/495(2006-01-01)

(21) (22)

Application

2004129725/04, 2003-03-04

(24)

Start date

2003-03-04

(22)

Actual filing date

2003-03-04

(45)

Published

2007-05-20

(72)

Inventor

Khajasi KazujaOdzima KatsudziKhori KozoOkudzo NorijukiMitsujama DzunitiKunitani KazutoTokhdo Kejsuke

(73)

Holder

Tojama Kemikal Ko., Ltd.

NOVEL DERIVATIVE OF ARYLAMIDINE OR ITS SALT Russian patent published in 2007 - IPC C07C257/18 C07D241/08 A61K31/155 A61K31/495

Abstract RU 2299195 C2

FIELD: organic chemistry, fungicides.

SUBSTANCE: invention relates to derivatives of arylamidine or its salts of the general formula (I): wherein X represents unsubstituted lower alkylene or alkenylene group or that substituted with hydroxy-group, alkyl or alkoxy-group; G¹ represents oxygen atom, sulfur atom or imino-group; G² represents carbon atom or nitrogen atom; R^a represents hydrogen atom, halogen atom and alkyl or alkoxy-group; R¹ represents unprotected or protected amidino-group or unsubstituted amidino-group or that substituted with hydroxy-group or alkyl; R² represents amino-substituted or substituted cyclic amino-group. Proposed compound possess the antifungal effect and high safety.

EFFECT: valuable biological properties of compounds.

10 cl, 14 tbl, 164 ex

Similar patents RU2299195C2

Title	Year	Author	Number
QUINOLONE COMPOUND AND PHARMACEUTICAL COMPOSITION	2009	Otsubo Kendzi Jamauti Takakhito Oti Judzi	RU2544530C2
NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVES, PHARMACEUTICAL COMPOSITION BASED ON SAID AND METHOD OF TREATMENT OR PROPHYLAXIS OF THROMBOTIC DISEASES	1995	Kijoaki Katano Sokiti Okhuti Tomoaki Miura Ejki Sitara Masaro Simidzu Kazue Jaegasi Naoto Okhkura Jasuko Isomura Khirojuki Iida Midori Isikava Kendzi Asai Emiko Khatsusiba	RU2156763C2
PIPERAZINE-SUBSTITUTED BENZOTHIOPHENES FOR TREATING PSYCHIATRIC DISORDERS	2006	Jamasita Khirosi Matsubara Dzun Osima Kunio Kuroda Khideaki Ito Nobuaki Mijamura Sin Simizu Satosi Tanaka Tatsuesi Takakhasi Kharuka	RU2402549C2
COMPOSITIONS, SYNTHESIS AND METHOD FOR USING ATYPICAL ANTIPSYCHOTIC DRUGS OF QUINOLINE	2008	Bkhat Laksminarajan Mokhapatra Prabkhu P. Bkhat Seema Rani	RU2497819C2
BASIC NON-PEPTIDE ANTAGONISTS OF BRADYKININE AND THEIR PHARMACEUTICAL COMPOSITIONS	2003	Kal'Vani Federiko Katrambone Fernando Felichetti Patritsija Finchem Kristofer Ingo Dzholitti Alessandro Maggi Karlo Al'Berto Kuartara Laura Rossi Kristina Terrachano Roza	RU2327688C2
1,2,5-THIADIAZOLE DERIVATIVES OF INDOLYLALKYL-PYRIMIDINYL-PIPERAZINES AND PHARMACEUTICAL COMPOSITION BASED ON THESE COMPOUNDS	1996	Ronni R. Krenshou Ehdvard Kh. Rudiger Dehvid V. Smit Karola Solomon Dzhozef Jevich	RU2165420C2
BENZENE DERIVATIVES	1994	Nobukhiro Okhi Tatsuja Kato Tomokazu Ozaki	RU2127254C1
COMPOUND WITH ANTI-CANCER ACTIVITY	2019	Uchida Kenji Kawai Ryohei Yamamoto Keisuke Kanai Toshimi Ikota Hideo Imaeda Takashi Yoshida Kei	RU2809763C2
COMPOUND CAPABLE OF BONDING WITH S1P RECEPTOR AND PHARMACEUTICAL APPLICATION THEREOF	2004	Nakade Sindzi Mizuno Khirotaka Ono Takedzi Minami Masasi Saga Khirosi Khagija Khirosi Komija Takaki Khabasita Khiromu Kurata Kharuto Okhtsuki Kazukhiro Kusumi Kensuke	RU2390519C2
4-AMINO-5-CYANOPYRIMIDINE DERIVATIVES	2005	Kato Masaja Sato Norifumi Okada Minoru Uno Tetsujuki Ito Nobuaki Takedzi Jasukhiro Sinokhara Khisasi Fuva Masakhiro	RU2386628C2

RU 2 299 195 C2

Authors

Khajasi Kazuja

Odzima Katsudzi

Khori Kozo

Okudzo Norijuki

Mitsujama Dzuniti

Kunitani Kazuto

Tokhdo Kejsuke

Dates

2007-05-20—Published

2003-03-04—Filed