COMPOUNDS, ACTIVE TOWARDS PPAR (PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR) Russian patent published in 2011 - IPC C07D409/14 C07D413/14 A61K31/405 A61P3/10 

Abstract RU 2419618 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a compound having structure

, radicals are as described in the formula of invention, as well as pharmaceutically-acceptable salt, prodrug, tautomer and stereoisomer thereof. The invention also relates to a composition, a set for modulating PPAR based on said compound, a method of treating a patient suffering from a disease or condition or at risk of a disease or condition, for which PPAR modulation is therapeutically useful.

EFFECT: novel compounds which are active towards PPAR are obtained and described.

41 cl, 622 ex, 8 tbl

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RU 2 419 618 C2

Authors

Lin Dzhek

Uomak Patrik

Li B'Jungkhun

Shi Shengkhua

Zhang Chao

Tsukerman Rebekka

Artis Din R.

Ibrakhim Prabkha N.

Vang Vejru

Dates

2011-05-27Published

2006-09-06Filed