COMBINATION CONTAINING N-METHOXY-3-METHYLPYRAZINE-2-YL)-2-(4-[1,3,4-OXADIAZOL-2-YL]PHENYL)PYRIDINE-3-SULFONAMIDE AND ANTIMITOTIC SUBSTANCE FOR MALIGNANT GROWTH Russian patent published in 2011 - IPC A61K31/497 A61P35/00 

Abstract RU 2428188 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to oncology, namely to agents for cancer treatment. The combination contains N-(3-methoxy-6-methylpyrazine-2-yl)-2-(4 -[1,3,4-oxadiazol-2-yl]phenyl)pyridine-3-sulfonamide and taxane or its derivatives, namely paclitaxel, docetaxel. The pharmaceutical composition contains such combinations in combination with one or more pharmaceutically acceptable diluents. Application of the combination for preparing the drug and treating or preventing cancer.

EFFECT: use of the combinations, the pharmaceutical composition allows providing higher clinical effectiveness.

12 cl, 6 ex, 3 dwg

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RU 2 428 188 C2

Authors

Bojl Fransis Tomas

Karuehn Dzhon

Kh'Juz Ehndr'Ju

Dzhonstoun Donna

Dates

2011-09-10Published

2005-11-23Filed