Show metadata Hide metadata

(19)

(11)

2 447 059

(13)

(51)

IPC

C07C231/04(2006-01-01)

C07C233/66(2006-01-01)

C07C233/92(2006-01-01)

A61P29/00(2006-01-01)

A61K31/167(2006-01-01)

(21) (22)

Application

2010130988/04, 2010-07-23

(24)

Start date

2010-07-23

(22)

Actual filing date

2010-07-23

(45)

Published

2012-04-10

(72)

Inventor

Vlasova Nadezhda AleksandrovnaKurbatov Evgenij RaisovichKorkodinova Ljubov' MikhajlovnaMardanova Ljudmila Gennad'EvnaShakirova Anzhelika Borisovna

(73)

Holder

Gosudarstvennoe Obrazovatel'Noe Uchrezhdenie Vysshego Professional'Nogo Obrazovanija Gosudarstvennaja Farmatsevticheskaja Akademija Federal'Nogo Agentstva Po Zdravookhraneniju I Sotsial'Nomu Razvitiju" Vpo Pgfa Roszdrava)Gosudarstvennoe Obrazovatel'Noe Uchrezhdenie Vysshego Professional'Nogo Obrazovanija Gosudarstvennyj Universitet" Vpo Pgu)

ANALGESIC AGENT Russian patent published in 2012 - IPC C07C231/04 C07C233/66 C07C233/92 A61P29/00 A61K31/167

Abstract RU 2447059 C2

FIELD: chemistry.

SUBSTANCE: invention relates to organic chemistry and specifically to novel compounds of the class of amides of NH-acyl-5-iodoanthranilic acid of general formula

where: R¹=CH₂C₆H₅, R=4-NO₂ (I); R¹=CH₂CH=CH₂, R=3-NO₂(II); R¹=CH₂CH=CH₂, R=4-CH₃ (III).

EFFECT: compounds have high analgesic activity and are virtually non-toxic.

1 cl, 6 ex, 1 tbl

Similar patents RU2447059C2

Title	Year	Author	Number
N-(4'-METHYLBENZOYL)-3,5-DICHLOROANTHRANILIC ACID BUTYLAMIDE EXHIBITING ANTI-INFLAMMATORY AND ANALGETIC ACTIVITY	2020	Andryukov Konstantin Vyacheslavovich Korkodinova Lyubov Mikhajlovna Rudakova Irina Pavlovna Chashchina Svetlana Viktorovna	RU2753655C1
METHYL AMIDE AND BENZYLAMIDE OF N-ACETYL-3,5-DIBROM-ANTHRANILIC ACID, DEMONSTRATING ANTI-INFLMAMMATORY AND ANALGETIC ACTIVITY	2007	Andrjukov Konstantin Vjacheslavovich Korkodinova Ljubov' Mikhajlovna Mardanova Ljudmila Gennad'Evna Vasil'Eva Marianna Jur'Evna	RU2342361C1
N-(2-FURANOYL)-5-IODOANTHRANYLIC ACID BENZYLAMIDE AND N-(2-FURANOYL)-5-IODOANTHRANYLIC ACID DIMETHYLAMIDE APPLICATION AS ANTIPHLOGISTIC MEDICINES	2006	Kurbatov Evgenij Raisovich Kurochkin Aleksej Viktorovich Korkodinova Ljubov' Mikhajlovna Syropjatov Boris Jakovlevich Markova Ljubov' Nikolaevna	RU2337101C1
METHOD FOR EXTRACTION OF ANALGETIC AGENTS	2011	Kurbatov Evgenij Raisovich Korkodinova Ljubov' Mikhajlovna Danilov Jurij Leonidovich Vakhrin Mikhail Ivanovich	RU2504771C2
4-METHYLPHENYLAMIDE N-BENZOYL-5-BROMO ANTHRANIC ACID WITH ANTI-INFLAMMATORY ACTIVITY	2017	Andryukov Konstantin Vyacheslavovich Korkodinova Lyubov Mikhajlovna Goldshtejn Aleksandr Grigorevich	RU2679892C1
2-{4-[2-(N,N-DIETHYLAMINO)ETHOXYCARBONYL]PHENYL} AMNO-4-OXO-4-R-PHENYL-2-BUTENOIC ACIDS HAVING ANALGESIC ACTIVITY	2009	Nekrasov Denis Denisovich Unizhuk Ekaterina Gennad'Evna Makhmudov Ramiz Ragibovich	RU2405767C1
DIARYLAMINES AND SYNTHESIS METHOD THEREOF	2010	Maslivets Andrej Nikolaevich Mashevskaja Irina Vladimirovna	RU2439053C1
ETHYL 1,6-DIARYL-4-AROYL-3-HYDROXY-2-OXO-8-PHENYL-1,7-DIAZASPIRO[4,4]NONA-3,6,8-TRIEN-9-CARBOXILATES AND METHOD OF THEIR OBTAINING	2011	Silajchev Pavel Sergeevich Makhmudov Ramiz Ragibovich Maslivets Andrej Nikolaevich	RU2467010C1
METHOD OF SELECTING ANTI-INFLAMMATORY AGENTS USING CALCULATED ENERGIES OF INTERACTION WITH ENZYMES CYCLOOXYGENASE 1 AND 2	2017	Andryukov Konstantin Vyacheslavovich Korkodinova Lyubov Mikhajlovna	RU2706366C2
DIMETHYL 2-ACYL-1-HYDROXY-3-METHYL-7-OXO-6-PHENYL-2,6-DIAZABICYCLO[3,2,1]OCT-3-ENE-5,8-DICARBOXYLATES AND METHOD FOR PREPARING THEM	2011	Silajchev Pavel Sergeevich Maslivets Andrej Nikolaevich Makhmudov Ramiz Ragibovich	RU2478638C1

RU 2 447 059 C2

Authors

Vlasova Nadezhda Aleksandrovna

Kurbatov Evgenij Raisovich

Korkodinova Ljubov' Mikhajlovna

Mardanova Ljudmila Gennad'Evna

Shakirova Anzhelika Borisovna

Dates

2012-04-10—Published

2010-07-23—Filed