NOVEL HETEROCYCLIDENE ACETAMIDE DERIVATIVE Russian patent published in 2012 - IPC C07D215/38 C07D215/08 C07D311/04 A61K31/4709 A61K31/353 A61P29/02 

Abstract RU 2451014 C2

FIELD: chemistry.

SUBSTANCE: invention relates to compounds of general formula

(where values of radicals are given in the claim), as well as salts of such compounds and pharmaceutical compositions based on such compounds. The described compounds exhibit type 1 channel antagonists with transient receptor potential (TRPV1).

EFFECT: compounds can be used to treat diseases and conditions causing pain.

30 cl, 255 ex, 40 tbl

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RU 2 451 014 C2

Authors

Utida Khidekharu

Kosuga Naoto

Satokh Tsutomu

Khotta Daido

Kamino Tomojuki

Maeda Jositaka

Amano Ken-Iti

Akada Jasusige

Dates

2012-05-20Published

2006-07-24Filed