COMBINATION OF IAP AND FLT3 INHIBITORS Russian patent published in 2012 - IPC A61K31/16 A61K31/427 A61K31/437 A61K31/553 A61K31/704 A61P35/00 

Abstract RU 2456983 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: present invention refers to pharmaceutics and medicine, and concerns a combination showing IAP inhibitor and FLT3 inhibitor activity containing (S)-N-((S)-1-cyclohexyl-2-{(S)-2-[4-(4-fluorobenzoyl)thiazol-2-yl]pyrrolidin-1-yl}-2-oxoethyl)-2-methylaminopropionamide, the compound of formula

, a method of treating of acute myeloid leukemia, applying said combination for treating acute myeloid leukemia and a commercial packing containing said combination.

EFFECT: composition shows high efficacy.

9 cl, 16 dwg, 16 ex

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RU 2 456 983 C2

Authors

Griffin Dzhejms Duglas

Zauehl Li

Dates

2012-07-27Published

2007-11-27Filed