NEW COMPOUNDS MIMETICS AND USING THEM Russian patent published in 2012 - IPC C07D487/04 A61K31/4985 A61K31/53 A61K35/02 

Abstract RU 2457210 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: there are described new compounds of general formula (I):

in the form of a separate stereoisomer or mixed stereoisomers or in the form of its pharmaceutically acceptable salt wherein R1 is indazolyl or substituted indazolyl; R6 is C6aryl or C6-12aryl substituted by halogen, hydroxy, cyano and C1-6alkoxy; or C6heterocyclyl containing 1-2 heteroatoms specified in nitrogen or oxygen; each X2 and X3 independently mean hydrogen, hydroxy or phosphate.

EFFECT: prepared compounds may be used for preparing a drug preparation for treating or preventing cancer, particularly acute myeloid leukemia.

6 cl, 6 tbl, 8 ex, 4 dwg

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RU 2 457 210 C2

Authors

Chung Dzae Uk

Dzung Khi-Kiung

Dzung Kiung-Jun

Dzeong Min-Vook

La Khiun-Dzu

Li Sang-Khak

Kim Khoe-Moon

Dates

2012-07-27Published

2008-10-15Filed