POLYMER COMPOSITIONS OF CETP INHIBITORS Russian patent published in 2012 - IPC A61K31/421 A61K9/16 A61P3/06 

Abstract RU 2457841 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention relates to pharmaceutical field and deals with perorally bioavailable pharmaceutical composition, which contains (a) CETP inhibiting compound, which has formula , or its pharmaceutically acceptable salt: (b) concentration-increasing polymer and (c) optionally one or more surface active substances. Invention also relates to application of said composition for production of medication, which increases level of HDL-cholesterol in patient.

EFFECT: invention provides compositions, which increase level of HDL-cholesterol and characterised by improved bioavailability in introduction to patient.

20 cl, 4 ex

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RU 2 457 841 C2

Authors

Girz Sara

Louindzher Majkl

Makkelvi Krehjg A.

Mejer Robert F.

Chzhan Dina

Dates

2012-08-10Published

2007-02-09Filed