PHARMACEUTICAL PREPARATION Russian patent published in 2021 - IPC C07D403/12 A61K31/506 A61K9/16 A61P31/10 

Abstract RU 2760681 C2

FIELD: pharmaceuticals.

SUBSTANCE: invention relates to pharmaceutical compositions containing particles produced by spray drying of 2-(1,5-dimethyl-3-phenyl-1H-pyrrol-2-yl)-N-(4-(4-(5-fluoropyrimidine-2-yl)piperazine-1-yl)phenyl)-2-oxacetamide particles, as well as an application of the pharmaceutical compositions for prevention or treatment of a fungal infection.

EFFECT: pharmaceutical compositions based on 2-(1,5-dimethyl-3-phenyl-1H-pyrrol-2-yl)-N-(4-(4-(5-fluoropyrimidine-2-yl)piperazine-1-yl)phenyl)-2-oxacetamide exhibiting antifungal properties are produced.

30 cl, 3 dwg, 1 tbl, 5 ex

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RU 2 760 681 C2

Authors

Lo Derek

Sajbli Grekhem Edvard Morris

Dates

2021-11-29Published

2017-05-25Filed