3-(2-BROMOPHENYL) AND 3-BENZYL-4,5,6,7-TETRAHYDROINDAZOLE HYDROCHLORIDES, ANTIMICROBIAL AGENT BASED THEREON Russian patent published in 2012 - IPC C07D231/56 A61K31/416 A61P31/04 

Abstract RU 2469027 C2

FIELD: chemistry.

SUBSTANCE: present invention relates to organic chemistry and specifically to novel biologically active indazole compounds: 3-(2-bromophenyl)-4,5,6,7-tetrahydroindazole hydrochloride (1a) and 3-benzyl-4,5,6,7-tetrahydroindazole hydrochloride (1b) of general formula: Ia, b (R=C6H4Br-2 (a), CH2C6H5 (b)). The invention also relates to an antimicrobial agent based on compounds of formula (1a) or (1b).

EFFECT: novel indazole derivatives having antibacterial activity are obtained.

2 cl, 1 tbl, 3 ex

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RU 2 469 027 C2

Authors

Pantjukhin Aleksej Aleksandrovich

Pershina Natal'Ja Nikolaevna

Mikhajlovskij Aleksandr Georgievich

Vikhareva Elena Vladimirovna

Aleksandrova Galina Arsent'Evna

Krylova Irina Olegovna

Makhmudov Ramiz Ragibovich

Dates

2012-12-10Published

2011-02-25Filed