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(19)

(11)

2 469 042

(13)

(51)

IPC

C07J43/00(2006-01-01)

A61K31/58(2006-01-01)

A61P35/00(2006-01-01)

A61P13/00(2006-01-01)

A61P5/32(2006-01-01)

(21) (22)

Application

2009114753/04, 2007-09-17

(24)

Start date

2007-09-17

(22)

Actual filing date

2007-09-17

(45)

Published

2012-12-10

(72)

Inventor

Messinger JozefShen UveKhuzen BettinaTole Genrikh-KhubertKoskimies PasiKallio Lila

(73)

Holder

Zol'Vaj Farmas'Jutiklz Gmbkh

THERAPEUTICALLY ACTIVE TRIAZOLES AND USE THEREOF Russian patent published in 2012 - IPC C07J43/00 A61K31/58 A61P35/00 A61P13/00 A61P5/32

Abstract RU 2469042 C2

FIELD: chemistry.

SUBSTANCE: invention relates to novel estratrien-triazoles of general formula (I), which are useful in therapy, especially in treating and/or preventing steroid hormone dependent disorders, preferably steroid hormone dependent diseases or disorders requiring the inhibition of 17β-hydroxysteroid dehydrogenase (17β-HSD) such as 17β-HSD type 1, type 2 or type 3 enzyme.

EFFECT: improved method.

21 cl

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RU 2 469 042 C2

Authors

Messinger Jozef

Shen Uve

Khuzen Bettina

Tole Genrikh-Khubert

Koskimies Pasi

Kallio Lila

Dates

2012-12-10—Published

2007-09-17—Filed