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(19)

(11)

2 430 917

(13)

(51)

IPC

C07D401/12(2006-01-01)

C07D401/14(2006-01-01)

C07D471/04(2006-01-01)

A61K31/4427(2006-01-01)

A61P9/00(2006-01-01)

(21) (22)

Application

2008148290/04, 2007-05-08

(24)

Start date

2007-05-08

(22)

Actual filing date

2007-05-08

(45)

Published

2011-10-10

(72)

Inventor

Kishida MasashiMatsuura NaokoImase KhidetomoIvaki JukiUmemura IchiroOkhmori OsamuKavakhara Ehjdzhi

(73)

Holder

Novartis Ag

BICYCLIC DERIVATIVES AS CEPT INHIBITORS Russian patent published in 2011 - IPC C07D401/12 C07D401/14 C07D471/04 A61K31/4427 A61P9/00

Abstract RU 2430917 C2

FIELD: chemistry.

SUBSTANCE: invention describes novel bicyclic derivatives of general formula (I)

(values of radicals are given in the description) and a pharmaceutical composition containing said derivatives, as well as use of said novel compounds to treat or inhibit symptomatic diseases where CEPT is involved, and a method of treating said diseases.

EFFECT: high efficiency of using compounds when treating diseases.

14 cl, 34 ex

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RU 2 430 917 C2

Authors

Kishida Masashi

Matsuura Naoko

Imase Khidetomo

Ivaki Juki

Umemura Ichiro

Okhmori Osamu

Kavakhara Ehjdzhi

Dates

2011-10-10—Published

2007-05-08—Filed