METHOD OF PRODUCING HETEROCYCLE-SUBSTITUTED PYRIDINE DERIVATIVES Russian patent published in 2013 - IPC C07D413/04 C07D413/14 C07D401/02 C07D401/04 A61K31/4439 A61K31/444 A61P31/10 

Abstract RU 2474581 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a method of producing heterocycle-substituted pyridine derivatives of general formula (I) by reacting a compound of general formula (III) with a compound of formula (II) in a solvent and in the presence of a catalyst based on palladium or a base, where R1, R2, X, Y, Q, A, Z, R, R3 and R4 are described in the claim.

EFFECT: method enables to obtain pyridine derivatives on an industrial scale.

7 cl, 27 ex

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RU 2 474 581 C2

Authors

Niidzima Dzun

Josizava Kazukhiro

Kosaka Juki

Abe Sinija

Dates

2013-02-10Published

2008-12-25Filed