DRUG CARRIER Russian patent published in 2013 - IPC A61K9/127 A61K47/18 A61K47/24 A61K47/34 A61K31/7088 

Abstract RU 2476204 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: group of inventions refers to pharmacology and concerns a circulating drug carrier. The carrier contains polyethylene glycol modified phospholipid presented by general formula or its pharmaceutically acceptable salt: wherein X represents as follows or ; and n represents an integer 30 to 150 wherein R1 represents a residue of saturated unbranched fatty acid having 17 to 22 carbon atoms, and 2-O-(2-diethylaminoethyl)carbamoyl-1,3-O-dioleoyl glycerol. Polyethylene glycol modified phospholipid is found in the amount of 30 wt % - 50 wt % of total weight of lipids in the carrier. What is also presented is a pharmaceutical composition containing the carrier described above and a drug.

EFFECT: group of inventions prolongs a circulation time and respectively improves the efficacy of the drug.

6 cl, 19 dwg, 5 tbl, 49 ex

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RU 2 476 204 C2

Authors

Sonoke Satoru

Ueda Tosikhiro

Dates

2013-02-27Published

2008-07-30Filed