FIELD: chemistry.
SUBSTANCE: invention relates to substituted N-phenyl-bipyrrolidine ureas of formula (I) ,
where values of R, R1, R2, R3, R4 and R5 are given in claim 1.
EFFECT: compounds are capable of binding with the H3 receptor, which enables use thereof to prepare a pharmaceutical composition and for diseases associated with the central nervous system.
10 cl, 36 ex
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Authors
Dates
2013-03-27—Published
2008-10-14—Filed