SUBSTITUTED N-PHENYL-BIPYRROLIDINE UREAS AND THERAPEUTIC USE THEREOF Russian patent published in 2013 - IPC C07D207/06 C07D403/04 C07D403/14 C07D409/12 C07D413/14 A61K31/4025 A61P25/00 

Abstract RU 2478094 C2

FIELD: chemistry.

SUBSTANCE: invention relates to substituted N-phenyl-bipyrrolidine ureas of formula (I) ,

where values of R, R1, R2, R3, R4 and R5 are given in claim 1.

EFFECT: compounds are capable of binding with the H3 receptor, which enables use thereof to prepare a pharmaceutical composition and for diseases associated with the central nervous system.

10 cl, 36 ex

Similar patents RU2478094C2

Title Year Author Number
SUBSTITUTED N-PHENYLBIPYRROLIDINE CARBOXAMIDES AND THERAPEUTIC USE THEREOF 2008
  • Chekhtizkij Verngard
  • Gao Chzhunli
  • Kherst Uill'Jam Dzh.
  • Shvink Lotar
  • Shtengelin Zigfrid
RU2477720C2
SUBSTITUTED N-PHENYLBIPYRROLIDINE CARBOXAMIDES AND THERAPEUTIC USE THEREOF 2008
  • Chekhtizkij Verngard
  • Gao Chzhunli
  • Kherst Vill'Jam Dzh.
  • Shvink Lotar
  • Shtengelin Zigfrid
RU2477719C2
SUBSTITUTED TETRAHYDROPYRANSPIROPYRROLIDINONE AND TETRAHYDROPYRANSPIROPIPERIDINONE, BASED ON THEM PHARMACEUTICAL COMPOSITION AND APPLICATION FOR THERAPEUTIC PURPOSES 2009
  • Gao Chzhunli
  • Khartung Rajan
  • Stefani Dehvid
RU2519778C2
SUBSTITUTED N-PHENYLPYRROLIDINYL METHYLPYRROLIDINE AMIDES AND THERAPEUTIC USE THEREOF AS MODULATORS OF HISTAMINE H3 RECEPTOR 2008
  • Chekhtizkij Verngard
  • Gao Chzhunli
  • Kherst Uill'Jam Dzh.
  • Shvink Lotar
  • Shtengelin Zigfrid
RU2477721C2
CYCLOPROPYLAMIDE DERIVATIVES AS N-HISTAMINE RECEPTOR MODULATORS 2007
  • Lju Khuatsin
  • Blehk Lorens A.
  • Bennani Jussef L.
  • Kauert Marlon D.
RU2449989C2
QUINAZOLINE DERIVATIVES FOR SLOWING DOWN GROWTH OF CANCER CELLS AND METHOD OF OBTAINING THEM 2005
  • Kham Jang Dzin
  • Gong Dzi Khieon
  • Cha Mi Jang
  • Kim Dzong Voo
  • Kim Maeng Sup
  • Kim Eun Jang
  • Song Dzi Jeon
  • Kim Chang In
  • Kim Se Jang
  • Li Gvan Sun
RU2362773C2
4-SUBSTITUTED-2-PHENOXYPHENYLAMINE MODULATORS OF DELTA-OPIOID RECEPTORS 2010
  • Kouts Stiven Dzh.
  • Bian Khajan
  • Tsaj Chaochzhun
  • De Kort Bart L.
  • Lju Li
  • Mehsilag Mark Dzh.
  • Daks Skott L.
  • Pitis Filip M.
  • Konnolli Piter Dzh.
  • Khe Vej
RU2553453C2
PYRROLE DERIVATIVES AS MEDICINAL SUBSTANCES 2005
  • Kanne Bannen Linn
  • Chen Dzheff
  • Dehlrimpl Liza Ehster
  • Flehtt Brenton T.
  • Forsajt Timoti Patrik
  • Gu Sjao-Khoj
  • Mehk Morrison B.
  • Mann Larri U.
  • Mann Grejs
  • Martin Richard
  • Mokhan Radzhu
  • Merfi Brehtt
  • Najman Majkl Charl'Z
  • Stivens Uill'Jam K. Ml.
  • Van Te-Lin'
  • Van Jun
  • Vu Dzhejson Kh.
RU2470916C2
PROTEIN TYROSINE KINASE ACTIVITY INHIBITORS 2009
  • Majkl Mannion
  • Stefan Rappel'
  • Stiven Uill'Jam Klaridzh
  • Frederik Godett
  • Litszi Chzhan'
  • Ljubomir Isakovits
  • Oskar Mario Saavedra
  • Tetsujuki Uno
  • Masashi Kishida
  • Arkadij Vajsburg
RU2533827C2
PYRIMIDINE AMIDE COMPOUNDS AS PGDS INHIBITORS 2006
  • Oldous S'Juzan S.
  • Tszjan' Dzhon Tszytsi
  • Lu Tszin'Tsi
  • Ma Ljan
  • Mu Lan'
  • Manson Khehrri Rendall
  • Sejbol Dzheffri Stefen
  • Tkhurajratnam Sukantkhini
  • Vandjuzen Kristofer Loren
RU2420519C2

RU 2 478 094 C2

Authors

Chekhtizkij Verngard

Gao Chzhunli

Kherst Uill'Jam Dzh.

Shvink Lotar

Shtengelin Zigfrid

Dates

2013-03-27Published

2008-10-14Filed