COMPOUNDS OF ((PHENYL)IMIDAZOLYL)METHYL-HETEROARYL, USE THEREOF, PHARMACEUTICAL COMPOSITION CONTAINING SAID COMPOUNDS, AND KIT CONTAINING SUCH COMPOSITION Russian patent published in 2013 - IPC C07D401/06 C07D409/06 A61K31/4178 A61P23/00 A61P29/00 

Abstract RU 2478631 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: present invention refers to new derivatives of ((phenyl)imidazolyl)methylheteroaryl of formula wherein A represents pyridyl or thienyl having 0 or 1 substitute; B represents phenyl having 0, 1 or 2 substitutes; wherein each substitute independently represents alkyl having 1 to 8 carbon atoms, -F, -Cl, -Br or -CF3. Also, the invention refers to the use of the declared compounds for the purpose of preparing a therapeutic agent, a pharmaceutical composition on the basis of the declared compounds, and to a kit containing the pharmaceutical composition above.

EFFECT: there are prepared new derivatives of ((phenyl)imidazolyl)methylheteroaryl effective in pain management.

10 cl, 1 tbl, 2 ex

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RU 2 478 631 C2

Authors

Sinkha Santosh S.

Khejdelbau Tod M.

Chou Ken

Bkheht Smita S.

Nguen Fong Kh.

Garst Majkl E.

Dates

2013-04-10Published

2008-05-13Filed