CHEMICAL METHOD Russian patent published in 2013 - IPC C07D209/08 C07C69/732 

Abstract RU 2481331 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a method of producing a compound of formula II from a compound of formula III: , where R1 and R2 are independently Cl, Br, F, I, via reaction thereof with an ester of formula (IV) , where R3 is C1-6alkyl; to obtain a compound of formula V: , which reacts with a hydroxyl ion in the presence of an aryl-alkyl ammonium salt or tetra-alkyl ammonium salt, to obtain a compound of formula VI , followed by treatment thereof to obtain a compound of formula VII: , which is reduced to obtain a compound of formula II.

EFFECT: high efficiency of the method.

5 cl, 9 ex

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RU 2 481 331 C2

Authors

Arnott Juan Aleksander

Krosbi Dzhon

Ehvans Matt'Ju Charlz

Ford Dzhejms Gejr

Dzhouns Martin Fransis

Lesli Kevin Uill'Jam

Makfarlejn Ajan Majkl

Sipenda Dzhordzh Dzhozef

Dates

2013-05-10Published

2007-11-01Filed