FIELD: chemistry.
SUBSTANCE: invention relates to a method for regioselective synthesis of 1-alkyl-3-halogenalkylpyrazole-4-carboxylic acid derivatives by reacting 2-acylated or 2-iminoalkylated acrylic acid derivative with N-alkylhydrazone, followed by cyclisation of the obtained intermediate compound. The invention also relates to an intermediate compound.
EFFECT: high regioselectivity of the method.
3 cl, 5 ex
Title | Year | Author | Number |
---|---|---|---|
METHOD FOR REGIOSELECTIVE SYNTHESIS OF 1-ALKYL-3-HALOGENALKYLPYRAZOLE-4-CARBOXYLIC ACID DERIVATIVES | 2013 |
|
RU2661192C2 |
METHOD FOR REGIOSELECTIVE SYNTHESIS OF 1-ALKYL-3-HALOGENALKYLPYRAZOLE-4-CARBOXYLIC ACID DERIVATIVES | 2009 |
|
RU2498978C2 |
METHOD OF PRODUCING 3-DIHALOMETHYL-PYRAZOLE-4-CARBOXYLIC ACID DERIVATIVES | 2007 |
|
RU2470015C2 |
SERINE-THREONINE PROTEIN KINASE AND PARP MODULATORS | 2013 |
|
RU2681209C2 |
DERIVATIVES OF INDOLE ORDER AS p38 KINASE INHIBITORS | 2000 |
|
RU2278115C2 |
HETEROARYL COMPOUNDS AS IRAK INHIBITORS AND USE THEREOF | 2016 |
|
RU2743360C2 |
HERBICIDAL COMPOSITION AND METHOD FOR WEED CONTROLLING | 1999 |
|
RU2261598C9 |
POLYMERISABLE UV AND HIGH ENERGY VISIBLE BLUE ABSORBERS | 2019 |
|
RU2796920C2 |
4-SUBSTITUTED PHENYLAMINE DERIVATIVES AND THEIR USE TO PROTECT CROPS AGAINST UNDESIRABLE PHYTOPATHOGENIC MICROORGANISMS | 2017 |
|
RU2796397C2 |
PYRAZOLOPYRIMIDINES AND RELATED HETEROCYCLES AS CK2 INHIBITORS | 2010 |
|
RU2607453C2 |
Authors
Dates
2013-11-20—Published
2009-02-12—Filed