METHOD FOR REGIOSELECTIVE SYNTHESIS OF 1-ALKYL-3-HALOGENALKYLPYRAZOLE-4-CARBOXYLIC ACID DERIVATIVES Russian patent published in 2013 - IPC C07D231/12 C07C251/76 C07C251/86 

Abstract RU 2498977 C9

FIELD: chemistry.

SUBSTANCE: invention relates to a method for regioselective synthesis of 1-alkyl-3-halogenalkylpyrazole-4-carboxylic acid derivatives by reacting 2-acylated or 2-iminoalkylated acrylic acid derivative with N-alkylhydrazone, followed by cyclisation of the obtained intermediate compound. The invention also relates to an intermediate compound.

EFFECT: high regioselectivity of the method.

3 cl, 5 ex

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RU 2 498 977 C9

Authors

Patsenok Sergij

Lui Norbert

Khajnrikh Jens-Ditmar

Voll'Ner Tomas

Dates

2013-11-20Published

2009-02-12Filed